SCHEMBL7790196

SCHEMBL7790196

O=C(NCc1ccncc1)Nc1ccccc1.O=C(O)C[C@@H](NC(=O)OCc1ccccc1)c1cccc(N=S(=O)=O)c1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.47
ITGB3 P05106 6/20 0.46
ITGAV P06756 6/20 0.46
NAMPT P43490 6/20 0.44
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7785616 0.92 NAMPT (0.49) ITGB3ITGAVNAMPT
SCHEMBL7790192 0.81 NAMPT (0.58) HTTITGB3ITGAVNAMPT
SCHEMBL7785608 0.73 NAMPT (0.57) ITGB3ITGAVNAMPT
SCHEMBL4955915 0.71 ITGB3 (0.43) HTTITGB3ITGAV
SCHEMBL6156731 0.70 CASP1 (0.60)
SCHEMBL6955527 0.70 CASP1 (0.60)
SCHEMBL6156740 0.70 CASP1 (0.60)
SCHEMBL7061672 0.69 PPARG (0.51)
SCHEMBL11616834 0.69 HTT (1.00) HTTNAMPTROCK2ROCK1POLB
SCHEMBL3857870 0.68 CASP1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147079-A2 BETA-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS Bayer Aktiengesellschaft (DE) 2001-10-24 EP disclosed
WO-2000041469-A2 β-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2000-07-20 WO disclosed