SCHEMBL7792606

SCHEMBL7792606

COc1ccc(CCN)cc1OC.O=C(O)c1ccc(Br)cc1.O=Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
ATM Q13315 1/20 0.45
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
MMP1 P03956 2/20 0.40
NR1H4 Q96RI1 1/20 0.40
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TSHR P16473 2/20 0.39
TAAR1 Q96RJ0 2/20 0.39
MAPK1 P28482 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4-Methylbenzoic Acid SCHEMBL7798453 0.91 KDM4E (0.46) KDM4EATMTDP1ALDH1A1MAPT
SCHEMBL7798405 0.90 SMN1; SMN2 (0.46) KDM4EATMTDP1ALDH1A1MAPT
SCHEMBL7798806 0.87 KDM4E (0.60) KDM4EATMTDP1ALDH1A1MMP1
SCHEMBL7798027 0.86 KDM4E (0.46) KDM4ETDP1ALDH1A1MAPTPPARD
Tyramine SCHEMBL8039128 0.84 SRD5A2 (0.41) KDM4ETDP1ALDH1A1L3MBTL1TAAR1
Phenethylamine SCHEMBL7799012 0.84 RXRA (0.42) ALDH1A1TAAR1RXRARXRBRXRG
SCHEMBL7798427 0.83 SRD5A2 (0.40) ATMALDH1A1MAPTTSHRTAAR1
SCHEMBL8037475 0.83 RXRA (0.44) PPARDPPARARXRARXRBRXRG
SCHEMBL7798600 0.82 SRD5A2 (0.46) RXRARXRBSMN1; SMN2
SCHEMBL7792608 0.82 HPGD (0.46) KDM4EALDH1A1MAPTRXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed