SCHEMBL7792608

SCHEMBL7792608

COc1ccc(C(C)N)cc1OC.O=C(O)c1ccc(Br)cc1.O=Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.46
AKR1C3 P42330 3/20 0.42
AKR1C2 P52895 3/20 0.42
ALDH1A1 P00352 2/20 0.41
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA7 P43166 1/20 0.39
TPMT P51580 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
ACHE P22303 1/20 0.38
POLB P06746 1/20 0.37
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
MAPT P10636 4/20 0.36
NPC1 O15118 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7798409 0.90 AKR1C3 (0.44) AKR1C3AKR1C2ALDH1A1CA12CA1
SCHEMBL7798808 0.87 ALDH1A1 (0.45) AKR1C3AKR1C2ALDH1A1CA1CA2
SCHEMBL7792606 0.82 KDM4E (0.45) ALDH1A1CA12CA1CA2CA4
SCHEMBL7792603 0.80 MAPT (0.44) HPGDALDH1A1CA12CA1CA2
4-Methylbenzoic Acid SCHEMBL7798453 0.73 KDM4E (0.46) ALDH1A1MAPTNPC1GAARAB9A
SCHEMBL7798027 0.72 KDM4E (0.46) AKR1C3ALDH1A1ACHEMAPTNPC1
SCHEMBL7798405 0.72 SMN1; SMN2 (0.46) ALDH1A1RXRARXRBRXRGMAPT
4-Methylbenzoic Acid SCHEMBL7798452 0.71 GAA (0.43) HPGDALDH1A1CA12CA1CA2
Phenethylamine SCHEMBL7799012 0.70 RXRA (0.42) ALDH1A1RXRARXRBRXRGNPC1
SCHEMBL7798400 0.70 HDAC1 (0.43) RXRARXRBRXRGMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed