SCHEMBL7794460

SCHEMBL7794460

CN(C)C(=O)Nc1ccccc1-c1ccc(CBr)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 1/20 0.48
GAA P10253 2/20 0.44
LMNA P02545 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 9/20 0.44
MAPT P10636 3/20 0.44
HTT P42858 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NPSR1 Q6W5P4 2/20 0.41
SOAT1 P35610 2/20 0.41
KCNQ2 O43526 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7795981 0.88 FABP4 (0.50) FABP4GAALMNAMEN1KMT2A
SCHEMBL10768865 0.83 FABP4 (0.64) FABP4MEN1KMT2AL3MBTL1ALDH1A1
SCHEMBL7791694 0.81 CHRM3 (0.45) GAALMNAMEN1KMT2AL3MBTL1
SCHEMBL7021257 0.79 MCL1 (0.38) FABP4GAALMNAMEN1KMT2A
SCHEMBL19181534 0.78 ALDH1A1 (0.49) FABP4GAALMNAMEN1KMT2A
SCHEMBL7089269 0.74 ALDH1A1 (0.56) ALDH1A1HTTKDM4E
SCHEMBL30761772 0.74 ALDH1A1 (0.56) ALDH1A1HTTKDM4E
SCHEMBL5105758 0.71 ALDH1A1 (0.56) GAALMNAMEN1KMT2AL3MBTL1
SCHEMBL10892045 0.70 ALDH1A1 (0.57) GAALMNAALDH1A1HTTMAPK1
SCHEMBL4139764 0.70 HTT (0.53) GAALMNAMEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0659179-B1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO INC (US) 2001-11-21 EP disclosed
US-5968924-A HAVE THE ABILITY TO STIMULATE THE RELEASE OF NATURAL OR ENDOGENOUS GROWTH HORMONE; TREATMENT OF OBESITY, OSTEOPOROSIS MERCK & CO., INC. (US) 1999-10-19 US disclosed
US-5672596-A ANIMAL GROWTH CONTROLLERS MERCK & CO., INC. (US) 1997-09-30 US disclosed
EP-0659179-A4 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE. MERCK & CO INC (US) 1995-08-09 EP disclosed
EP-0659179-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO. INC. (US) 1995-06-28 EP disclosed
WO-1994005634-A1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO., INC. (US) 1994-03-17 WO disclosed
US-5283241-A Animal growth regulators MERCK & CO., INC. (US) 1994-02-01 US disclosed