SCHEMBL7794523

SCHEMBL7794523

Cc1ccc([N]C2CCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 2/20 0.37
HTR3B O95264 2/20 0.37
HTR3A P46098 2/20 0.37
HTR3D Q70Z44 2/20 0.37
HTR3C Q8WXA8 2/20 0.37
SLC22A2 O15244 1/20 0.37
SLC22A1 O15245 1/20 0.37
SLC22A3 O75751 1/20 0.37
PLAU P00749 1/20 0.37
ACHE P22303 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
ALDH1A1 P00352 3/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SLC18A3 Q16572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2478208 0.95 CYP1A2 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7794041 0.93 NPC1 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7784569 0.91 ACHE (0.40) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7793278 0.83 HTR3E (0.34) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7793328 0.81 HTR3E (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7418307 0.73 SLC22A2 (0.37) SLC22A2SLC22A1SLC22A3PLAUTDP1
SCHEMBL7794037 0.72 CA12 (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL3146112 0.71 ALDH1A1 (0.39) ALDH1A1MEN1KMT2ASLC18A3TSHR
SCHEMBL7793271 0.71 SLC18A3 (0.46) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL723225 0.70 ALDH1A1 (0.39) ALDH1A1KMT2ASLC18A3MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed