SCHEMBL7794037

SCHEMBL7794037

COc1ccc([N]C2CCCC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
NOS3 P29474 2/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
KDM4E B2RXH2 2/20 0.41
SLC18A3 Q16572 1/20 0.41
RAB9A P51151 4/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790490 0.83 NOS3 (0.43) CA12CA1CA2CA7CA9
SCHEMBL2478208 0.77 CYP1A2 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7794041 0.75 NPC1 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7418307 0.72 SLC22A2 (0.37) NOS3RAB9AMEN1LMNAMAPT
SCHEMBL7794523 0.72 HTR3E (0.37) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL1129966 0.72 KMT2A (0.59) CA12CA2CA9RAB9ALMNA
SCHEMBL1129964 0.72 KMT2A (0.59) CA12CA2CA9RAB9ALMNA
SCHEMBL3146112 0.72 ALDH1A1 (0.39) SLC18A3MEN1KMT2ATSHRGAA
SCHEMBL19233521 0.71 KMT2A (0.62) CA12CA2CA9RAB9ALMNA
SCHEMBL22340416 0.71 GFER (0.48) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed