SCHEMBL7796696

SCHEMBL7796696

Cc1ccccc1C(=O)N1CCC2(CC1)N=C(N)c1ccccc1N2

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 8/20 0.48
NOS1 P29475 5/20 0.48
NOS3 P29474 2/20 0.48
HTT P42858 2/20 0.47
ABL1 P00519 1/20 0.46
BCR P11274 1/20 0.46
ALDH1A1 P00352 2/20 0.44
CCR5 P51681 1/20 0.41
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8376505 0.99 NOS2 (0.47) NOS2NOS1NOS3HTTABL1
SCHEMBL7806855 0.84 NOS2 (0.51) NOS2NOS1NOS3ABL1BCR
SCHEMBL7806816 0.84 NOS2 (0.56) NOS2NOS1NOS3ABL1BCR
SCHEMBL7804452 0.84 NOS2 (0.57) NOS2NOS1NOS3ALDH1A1
SCHEMBL7803469 0.83 NOS2 (0.50) NOS2NOS1NOS3ALDH1A1
Hydrochloric Acid SCHEMBL8379564 0.83 NOS2 (0.55) NOS2NOS1NOS3ABL1BCR
Hydrochloric Acid SCHEMBL8381626 0.83 NOS2 (0.50) NOS2NOS1NOS3ABL1BCR
SCHEMBL7802976 0.83 CA12 (0.46) NOS2NOS1NOS3HTTMAPT
Hydrochloric Acid SCHEMBL8378262 0.83 NOS2 (0.56) NOS2NOS1NOS3ALDH1A1
SCHEMBL7802914 0.83 GABRD (0.53) NOS2NOS1NOS3ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
EP-1100505-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR AstraZeneca AB (SE) 2001-05-23 EP claimed
WO-2000000200-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR ASTRAZENECA AB (SE) 2000-01-06 WO claimed