SCHEMBL7802976

SCHEMBL7802976

NC1=NC2(CCN(C(=O)c3ccccc3[N+](=O)[O-])CC2)Nc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
HPGD P15428 1/20 0.44
NOS2 P35228 5/20 0.43
NOS1 P29475 4/20 0.43
HTT P42858 2/20 0.43
LMNA P02545 1/20 0.43
MGLL Q99685 1/20 0.41
NOS3 P29474 1/20 0.41
PARP1 P09874 1/20 0.40
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8382208 0.99 CA12 (0.45) CA12CA1CA2CA7CA9
SCHEMBL7940838 0.84 NOS1 (0.52) CA12CA1CA2CA7CA9
SCHEMBL7796696 0.83 NOS2 (0.48) NOS2NOS1HTTNOS3MAPT
Hydrochloric Acid SCHEMBL8376562 0.83 NOS1 (0.52) CA12CA1CA2CA7CA9
Hydrochloric Acid SCHEMBL8376505 0.82 NOS2 (0.47) NOS2NOS1HTTNOS3MAPT
SCHEMBL7804502 0.82 RXFP1 (0.53) CA12CA1CA2CA7CA9
Hydrochloric Acid SCHEMBL8376490 0.81 RXFP1 (0.52) CA12CA1CA2CA7CA9
Hydrochloric Acid SCHEMBL8378262 0.79 NOS2 (0.56) HPGDNOS2NOS1NOS3
SCHEMBL7943022 0.79 NOS2 (0.48) HPGDNOS2NOS1HTTNOS3
SCHEMBL7803377 0.78 NOS2 (0.55) HPGDNOS2NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
EP-1100505-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR AstraZeneca AB (SE) 2001-05-23 EP claimed
WO-2000000200-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR ASTRAZENECA AB (SE) 2000-01-06 WO claimed