SCHEMBL7797244

SCHEMBL7797244

COc1ccccc1N1CC(c2ccccc2)OC1=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 5/20 0.61
ALDH1A1 P00352 2/20 0.47
POLB P06746 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HTR6 P50406 2/20 0.45
MAPK1 P28482 1/20 0.45
HSD11B1 P28845 2/20 0.45
ATM Q13315 1/20 0.44
ROCK2 O75116 1/20 0.44
ROCK1 Q13464 1/20 0.44
ADRA1D P25100 2/20 0.42
ADRA1A P35348 2/20 0.42
ADRA1B P35368 2/20 0.42
MGLL Q99685 1/20 0.42
ABCB1 P08183 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7944255 0.80 FADS1 (0.45) FADS1ALDH1A1KDM4EHTR6HSD11B1
SCHEMBL7807351 0.80 FADS1 (0.55) FADS1HSD17B10MEN1KMT2AHTR6
SCHEMBL27742774 0.80 ALDH1A1 (0.46) FADS1ALDH1A1POLBMEN1KMT2A
SCHEMBL7776725 0.78 FADS1 (0.60) FADS1ALDH1A1MEN1KMT2AHTR6
SCHEMBL19338270 0.78 GRM2 (0.47) FADS1ALDH1A1POLBMEN1KMT2A
SCHEMBL28922760 0.77 GRM2 (0.46) FADS1ALDH1A1POLBMEN1KMT2A
SCHEMBL9016279 0.76 FADS1 (0.79) FADS1HTR6HSD11B1ROCK2ROCK1
SCHEMBL7805542 0.75 HTR6 (0.65) FADS1HTR6HSD11B1
SCHEMBL7364885 0.71 FADS1 (0.50) FADS1KDM4EHSD17B10HTR6HSD11B1
SCHEMBL7364886 0.71 FADS1 (0.50) FADS1KDM4EHSD17B10HTR6HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255327-B1 ANTIHYPOXC, ANTIISCHEMIC AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-03 US disclosed
EP-1071670-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM KG (DE) 2001-01-31 EP disclosed
WO-1999054314-A1 NOVEL DIPHENYL-SUBSTITUTED 5-RING-HETEROCYCLES, METHOD FOR PRODUCING THEM AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-28 WO disclosed