SCHEMBL12963699

SCHEMBL12963699

CCCNc1cc(C)cc(C)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.55
NOS2 P35228 2/20 0.55
TLR8 Q9NR97 1/20 0.50
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
ALDH1A1 P00352 3/20 0.42
TP53 P04637 2/20 0.42
MAPK1 P28482 2/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
DNM2 P50570 6/20 0.41
LCK P06239 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
IDH1 O75874 1/20 0.39
NOS1 P29475 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9313985 0.89 TLR8 (0.65) NOS3NOS2TLR8ESR1ESR2
SCHEMBL24672584 0.87 TLR8 (0.58) NOS3NOS2TLR8ESR1ESR2
SCHEMBL8543215 0.85 DNM2 (0.57) NOS3NOS2TLR8ESR1ESR2
SCHEMBL8345724 0.83 NOS3 (0.59) NOS3NOS2TLR8ALDH1A1TP53
SCHEMBL11446300 0.83 NOS3 (0.46) NOS3NOS2TLR8ALDH1A1TP53
SCHEMBL7797450 0.82 NOS3 (0.53) NOS3NOS2TLR8ALDH1A1TP53
SCHEMBL23482212 0.82 GAA (0.56) NOS3NOS2TLR8ALDH1A1TP53
SCHEMBL11448132 0.80 NOS3 (0.47) NOS3NOS2TLR8ALDH1A1TP53
SCHEMBL11187910 0.79 DNM2 (0.55) NOS3NOS2TLR8ALDH1A1TP53
SCHEMBL16608745 0.78 DNM2 (0.61) TLR8ESR1ESR2ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7868204-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2011-01-11 US disclosed
US-7838520-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2010-11-23 US disclosed
US-7595343-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2009-09-29 US disclosed