SCHEMBL7799013

SCHEMBL7799013

C=CC(Cc1ccccc1)NC(=O)C(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CTRB1 P17538 4/20 0.44
POLB P06746 2/20 0.44
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
ALDH1A1 P00352 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
TSHR P16473 1/20 0.42
MME P08473 1/20 0.42
ACE P12821 1/20 0.42
ACE2 Q9BYF1 1/20 0.42
MAPK1 P28482 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6444347 0.85 CPA1 (0.44) CTSBNPC1RAB9ACTRB1NPSR1
SCHEMBL6981307 0.85 CTSB (0.43) CTSBNPC1RAB9ACTRB1ALDH1A1
SCHEMBL6444348 0.85 CPA1 (0.44) CTSBNPC1RAB9ACTRB1NPSR1
SCHEMBL7796543 0.83 CTRB1 (0.59) NPC1RAB9ACTRB1TAAR1
SCHEMBL28055494 0.83 CTRB1 (0.59) NPC1RAB9ACTRB1TAAR1
SCHEMBL3554246 0.82 CTRB1 (0.50) NPC1RAB9ACTRB1TAAR1CYP1A2
SCHEMBL7626858 0.82 CTRB1 (0.50) NPC1RAB9ACTRB1TAAR1CYP1A2
SCHEMBL27809899 0.81 CAPN1 (0.46) CTSBNPC1RAB9ACTRB1CYP3A4
SCHEMBL5732519 0.81 ATM (0.57) CTSBALDH1A1ACE
SCHEMBL13937947 0.81 ATM (0.57) CTSBALDH1A1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748801-B1 2-ISOXAZOLINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING RELATED DERIVATIVES FROM THE SAME DAICEL CHEM (JP) 2001-12-19 EP disclosed
US-6018069-A 2-isoxazoline derivative and process for producing the same and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2000-01-25 US disclosed
US-5994558-A 2-isoxazoline derivative and process for producing the same; and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-30 US disclosed
US-5962692-A 2-isoxazoline derivative and process for producing the same, and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-05 US disclosed
US-5750717-A 2-isoxazoline derivative and process for producing the same, and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-12 US disclosed
EP-0748801-A1 2-ISOXAZOLINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING RELATED DERIVATIVES FROM THE SAME DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-18 EP disclosed