SCHEMBL3554246

SCHEMBL3554246

C=C[C@H](Cc1ccccc1)NC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 8/20 0.50
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
CAPN1 P07384 2/20 0.46
CYP1A2 P05177 1/20 0.46
PSMB8 P28062 1/20 0.45
PSMB5 P28074 1/20 0.45
ACE P12821 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
ALPI P09923 1/20 0.43
PKM P14618 1/20 0.43
PTGS1 P23219 1/20 0.43
XIAP P98170 1/20 0.43
SLC7A5 Q01650 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7626858 1.00 CTRB1 (0.50) CTRB1NPC1RAB9ACAPN1CYP1A2
SCHEMBL28055494 0.86 CTRB1 (0.59) CTRB1NPC1RAB9ATAAR1ALPI
SCHEMBL7796543 0.86 CTRB1 (0.59) CTRB1NPC1RAB9ATAAR1ALPI
SCHEMBL27809899 0.85 CAPN1 (0.46) CTRB1NPC1RAB9ACAPN1CYP1A2
SCHEMBL7796605 0.85 PSMB8 (0.56) PSMB8PSMB5
SCHEMBL7796444 0.85 CTRB1 (0.56) CTRB1NPC1RAB9ACAPN1ACE
SCHEMBL17865652 0.84 CAPN1 (0.61) CAPN1ACE
SCHEMBL3292711 0.84 CAPN1 (0.61) CAPN1ACE
SCHEMBL2369340 0.84 CAPN1 (0.61) CAPN1ACE
SCHEMBL7796647 0.83 CTSK (0.47) CTRB1NPC1RAB9ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697348-B1 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LAB (US) 2011-12-28 EP disclosed
US-7696226-B2 HIV protease inhibiting compounds ABBOTT LABORATORIES (US) 2010-04-13 US disclosed
US-20050159469-A1 HIV protease inhibiting compounds ABBVIE INC. 2005-07-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050159469-A1 HIV protease inhibiting compounds SERPINB1, HPN, DNPEP CTRB1 168/4885NPC1 569/4885RAB9A 2012/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.