SCHEMBL7800949

SCHEMBL7800949

CC(C)(C)OC(=O)NCCCC(=O)Cc1cccc(OCc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
SIGMAR1 Q99720 1/20 0.46
LTB4R Q15722 1/20 0.46
LTB4R2 Q9NPC1 1/20 0.46
MAOB P27338 1/20 0.44
HTT P42858 1/20 0.44
SYK P43405 1/20 0.44
CYP2D6 P10635 1/20 0.44
SPHK2 Q9NRA0 2/20 0.44
SPHK1 Q9NYA1 1/20 0.44
FFAR1 O14842 1/20 0.44
PDK1 Q15118 1/20 0.43
PDK2 Q15119 1/20 0.43
PDK3 Q15120 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7796788 0.87 HDAC3 (0.44) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL1295547 0.87 LTB4R (0.49) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL7281204 0.86 CYP2D6 (0.52) SIGMAR1MAOBCYP2D6
SCHEMBL24310073 0.85 PTPN1 (0.55) SIGMAR1MAOBSPHK2SPHK1NR4A2
SCHEMBL3715955 0.85 SIGMAR1 (0.56) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL31506266 0.84 CYP2D6 (0.58) LTB4RLTB4R2MAOBHTTCYP2D6
SCHEMBL67569 0.84 CYP2D6 (0.58) LTB4RLTB4R2MAOBHTTCYP2D6
SCHEMBL18551719 0.81 CA12 (0.53) PDK2IDO1
SCHEMBL26197202 0.80 LTB4R (0.51) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL32665611 0.79 SMPD1 (0.60) MAOBCYP2D6SPHK2SPHK1NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159260-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000055124-A2 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed