SCHEMBL7796788

SCHEMBL7796788

CC(CCC(=O)NCCCC(=O)Cc1cccc(OCc2ccccc2)c1)CNC(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
SYK P43405 1/20 0.43
LTA4H P09960 2/20 0.41
PSMB1 P20618 2/20 0.39
PSMB5 P28074 2/20 0.39
PSMB2 P49721 2/20 0.39
SIGMAR1 Q99720 1/20 0.39
HPGD P15428 2/20 0.39
PTGES O14684 1/20 0.39
VNN1 O95497 1/20 0.39
LTB4R Q15722 1/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
MME P08473 1/20 0.38
ACE P12821 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7800949 0.87 HDAC3 (0.48) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL7790129 0.83 CA1 (0.38) SYKSIGMAR1
SCHEMBL1295547 0.77 LTB4R (0.49) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL7281204 0.75 CYP2D6 (0.52) SIGMAR1
SCHEMBL7799740 0.74 SYK (0.47) SYKLTA4HSIGMAR1ACEMAPT
SCHEMBL24310073 0.74 PTPN1 (0.55) SIGMAR1
SCHEMBL3715955 0.74 SIGMAR1 (0.56) HDAC3HDAC1HDAC2HDAC10HDAC11
SCHEMBL31506266 0.73 CYP2D6 (0.58) LTA4HHPGDLTB4RLTB4R2
SCHEMBL67569 0.73 CYP2D6 (0.58) LTA4HHPGDLTB4RLTB4R2
SCHEMBL26197202 0.73 LTB4R (0.51) HDAC3HDAC1HDAC2HDAC10HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159260-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000055124-A2 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed