SCHEMBL7801432

SCHEMBL7801432

COc1ccc(CN2CCC(CCN)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.56
ACHE P22303 2/20 0.55
BACE1 P56817 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
MAOB P27338 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29201740 0.85 ACHE (0.62) SIGMAR1ACHEBACE1SMN1; SMN2MAOB
SCHEMBL13596996 0.84 MEN1 (0.57) SIGMAR1ACHEBACE1SMN1; SMN2MAOB
SCHEMBL8825661 0.83 SIGMAR1 (0.62) SIGMAR1ACHE
SCHEMBL15933891 0.83 ALDH1A1 (0.53) ACHEBACE1MAOBMEN1KMT2A
SCHEMBL621695 0.82 HRH3 (0.62) SIGMAR1ACHEBACE1SMN1; SMN2MEN1
SCHEMBL1586714 0.81 SIGMAR1 (0.63) SIGMAR1ACHEBACE1SMN1; SMN2MEN1
SCHEMBL8101249 0.81 SIGMAR1 (0.63) SIGMAR1ACHEBACE1SMN1; SMN2MEN1
Hydrochloric Acid SCHEMBL11534460 0.80 SIGMAR1 (0.61) SIGMAR1ACHEBACE1SMN1; SMN2MEN1
SCHEMBL8825473 0.80 SLC6A3 (0.56)
SCHEMBL8320248 0.80 HRH3 (0.69) SIGMAR1ACHEBACE1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673927-B1 piperidines as anticholinergic agents EISAI CO LTD (JP) 2001-09-19 EP disclosed
EP-1116716-A1 Piperidine and piperazine compounds for use in the treatment of Alzheimer Eisai Co., Ltd. (JP) 2001-07-18 EP disclosed
EP-0742207-A1 2-(Indan-1-one-2-yl-alkyl)-1-phenylalkyl-piperidines and processes for their preparation Eisai Co., Ltd. (JP) 1996-11-13 EP disclosed
EP-0673927-A1 4-[2-indanyl-1-one]alkylpiperidines as anticholinergic agents Eisai Co., Ltd. (JP) 1995-09-27 EP disclosed
EP-0579263-A1 1,4-Substituted piperidines as acetylchozinesterase inhibitors and their use for the treatment of Alzheimer's disease Eisai Co., Ltd. (JP) 1994-01-19 EP disclosed
US-5100901-A Treatment of Alzheimer*s disease EISAI CO., LTD. (JP) 1992-03-31 US disclosed
US-4895841-A Cyclic amine compounds with activity against acetylcholinesterase EISAI CO., LTD. (JP) 1990-01-23 US disclosed
EP-0296560-A2 1,4-Substituted piperidines as acetylcholinesterase inhibitors and their use for the treatment of Alzheimer's disease Eisai Co., Ltd. (JP) 1988-12-28 EP disclosed