SCHEMBL7802852

SCHEMBL7802852

CN(C(=O)CC(CCN1CCN(Cc2ccccc2)CC1)c1ccccc1)c1ccc(Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.62
CCR5 P51681 3/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
HTR7 P34969 1/20 0.46
SIGMAR1 Q99720 2/20 0.46
OPRM1 P35372 1/20 0.46
CACNA1G O43497 1/20 0.44
POLB P06746 1/20 0.44
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43
CACNA2D1 P54289 1/20 0.43
CACNA1B Q00975 1/20 0.43
CACNB1 Q02641 1/20 0.43
CACNA1C Q13936 1/20 0.43
FAAH O00519 2/20 0.43
ATM Q13315 2/20 0.43
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7807754 0.94 DRD4 (0.58) DRD4CCR5MEN1KMT2AHTR7
SCHEMBL7802841 0.84 OPRM1 (0.59) DRD4MEN1KMT2ASIGMAR1OPRM1
SCHEMBL7811493 0.80 TACR2 (0.57) DRD4CCR5OPRM1POLB
SCHEMBL7807765 0.80 DRD4 (0.46) DRD4MEN1KMT2ACACNA2D1CACNA1B
SCHEMBL7815183 0.79 TACR2 (0.56) CCR5
SCHEMBL7812086 0.77 GABBR2 (0.50) DRD4MEN1KMT2APOLB
SCHEMBL7802957 0.76 TACR2 (0.66) OPRM1
SCHEMBL7802820 0.76 OPRL1 (0.58) OPRM1KDM4E
SCHEMBL7815271 0.76 TACR2 (0.48)
SCHEMBL7807766 0.73 DRD4 (0.41) DRD4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-B1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2001-10-31 EP disclosed
US-5654316-A Piperidine derivatives as neurokinin antagonists SCHERING CORPORATION (US) 1997-08-05 US disclosed