SCHEMBL7804223

SCHEMBL7804223

COC(=O)CC(Cc1ccc(O)cc1)c1ncc(C)s1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSA P10619 16/20 0.42
ESR1 P03372 2/20 0.40
ESR2 Q92731 2/20 0.40
PTGS2 P35354 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6493992 0.86 CTSA (0.46) CTSA
SCHEMBL27510388 0.86 MAOB (0.53) CTSA
SCHEMBL27535196 0.79 ESR1 (0.41) CTSAESR1ESR2
SCHEMBL6504253 0.76 ITGB3 (0.61)
SCHEMBL6499973 0.74 PKM (0.51) CTSA
SCHEMBL7259084 0.72 ESR1 (0.50) ESR1ESR2
SCHEMBL7803616 0.72 ESR1 (0.37) ESR1ESR2PTGS2
SCHEMBL27557934 0.72 ESR1 (0.41) CTSAESR1ESR2
SCHEMBL27535182 0.71 ESR1 (0.52) ESR1ESR2
SCHEMBL27535185 0.71 ESR1 (0.43) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1236767-C Vitronectin receptor antagonists SMITHKLINE BEECHAM CORP (US) 2006-01-18 CN disclosed
US-6881736-B1 Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2005-04-19 US disclosed
US-6881736-B1 Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2005-04-19 US disclosed
CN-1377269-A Vitronectin receptor antagonists SMITHKLINE BEECHAM CORP (US) 2002-10-30 CN disclosed