SCHEMBL7805028

SCHEMBL7805028

NC1=NC2(CCN(C(=O)c3ccc(Cl)cc3)CC2)Nc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 7/20 0.56
NOS1 P29475 6/20 0.56
IP6K1 Q92551 3/20 0.49
IP6K3 Q96PC2 1/20 0.49
IP6K2 Q9UHH9 1/20 0.49
ABL1 P00519 2/20 0.47
BCR P11274 2/20 0.47
HTR1A P08908 1/20 0.46
HTR2A P28223 1/20 0.46
HTR7 P34969 1/20 0.46
HTR6 P50406 1/20 0.46
NEK2 P51955 1/20 0.46
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
KCNH2 Q12809 2/20 0.43
NOS3 P29474 1/20 0.43
CCR8 P51685 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8381634 0.99 NOS2 (0.55) NOS2NOS1IP6K1IP6K3IP6K2
Trifluoroacetic Acid SCHEMBL7975720 0.93 NOS2 (0.52) NOS2NOS1IP6K1IP6K3IP6K2
SCHEMBL7796711 0.91 NOS2 (0.58) NOS2NOS1IP6K1IP6K3IP6K2
SCHEMBL7804452 0.91 NOS2 (0.57) NOS2NOS1NEK2ALDH1A1LMNA
SCHEMBL7931778 0.90 NOS2 (0.57) NOS2NOS1IP6K1IP6K3IP6K2
Hydrochloric Acid SCHEMBL8379932 0.90 NOS2 (0.57) NOS2NOS1IP6K1IP6K3IP6K2
SCHEMBL7796668 0.90 NOS2 (0.57) NOS2NOS1IP6K1IP6K3IP6K2
Hydrochloric Acid SCHEMBL8378262 0.90 NOS2 (0.56) NOS2NOS1NEK2ALDH1A1KCNH2
SCHEMBL7802943 0.89 NOS2 (0.61) NOS2NOS1ABL1BCRNEK2
Hydrochloric Acid SCHEMBL8376965 0.89 NOS2 (0.56) NOS2NOS1IP6K1IP6K3IP6K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
EP-1100505-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR AstraZeneca AB (SE) 2001-05-23 EP claimed
WO-2000000200-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR ASTRAZENECA AB (SE) 2000-01-06 WO claimed