SCHEMBL195205

SCHEMBL195205

NS(=O)(=O)NCC1CC(S)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
RAB9A P51151 4/20 0.38
ALDH1A1 P00352 2/20 0.38
DPP8 Q6V1X1 1/20 0.38
DPP9 Q86TI2 1/20 0.38
MAPT P10636 3/20 0.38
NPC1 O15118 2/20 0.38
ATM Q13315 1/20 0.38
HPGD P15428 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
IDO1 P14902 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL195204 1.00 CA12 (0.40) CA12CA1CA2CA7CA9
SCHEMBL9519385 0.90 ALDH1A1 (0.40) TDP1ALDH1A1MAPTATMHPGD
SCHEMBL7805565 0.85 CA12 (0.41) CA12CA1CA2CA9ALDH1A1
SCHEMBL7811546 0.84 RAB9A (0.43) TDP1RAB9AALDH1A1DPP8DPP9
SCHEMBL10364355 0.83 TDP1 (0.43) TDP1RAB9AALDH1A1MAPTNPC1
SCHEMBL6398540 0.83 TDP1 (0.43) TDP1RAB9AALDH1A1MAPTNPC1
SCHEMBL8759638 0.83 TDP1 (0.43) TDP1RAB9AALDH1A1MAPTNPC1
SCHEMBL10370030 0.83 RAB9A (0.42) TDP1RAB9AALDH1A1DPP8DPP9
SCHEMBL7811544 0.82 CCR5 (0.41) TDP1RAB9AMAPTNPC1ATM
SCHEMBL10370916 0.82 RAB9A (0.42) TDP1RAB9AALDH1A1DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012114280-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF PYRROLIDINE THIOL DERIVATIVES USEFUL IN THE SYNTHESIS OF CARBAPENEM COMPOUNDS ORCHID CHEMICALS AND PHARMACEUTICALS LIMITED (IN) 2012-08-30 WO disclosed
EP-2401278-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF CARBAPENEM ANTIBIOTIC Orchid Chemicals&Pharmaceuticals Limited (IN) 2012-01-04 EP disclosed
WO-2010097686-A1 AN IMPROVED PROCESS FOR THE PREPARATION OF CARBAPENEM ANTIBIOTIC ORCHID CHEMICALS & PHARMACEUTICALS LTD (IN) 2010-09-02 WO disclosed
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed