SCHEMBL7809178

SCHEMBL7809178

COc1ccc(COC(=O)N2C[C@H](OS(C)(=O)=O)C[C@H]2CNS(N)(=O)=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA5A P35218 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
GRIN2B Q13224 1/20 0.38
HTT P42858 2/20 0.38
PKM P14618 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MMP1 P03956 2/20 0.38
MMP3 P08254 2/20 0.38
MMP7 P09237 2/20 0.38
MMP9 P14780 2/20 0.38
MMP13 P45452 1/20 0.38
ITGB3 P05106 3/20 0.37
ITGB1 P05556 3/20 0.37
ITGAV P06756 3/20 0.37
ITGA5 P08648 3/20 0.37
ITGB5 P18084 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7806890 0.88 CA12 (0.42) CA12CA1CA2CA5ACA9
SCHEMBL7811567 0.86 PKM (0.39) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7805565 0.85 CA12 (0.41) CA12CA1CA2CA5ACA9
SCHEMBL7809302 0.82 CA12 (0.38) CA12CA1CA2CA5ACA9
SCHEMBL9428692 0.81 MMP2 (0.50) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7805540 0.81 MMP2 (0.50) GRIN2BHTTPKMSMN1; SMN2MMP1
SCHEMBL7805526 0.79 CASP3 (0.41) GRIN2BHTTMMP1MMP3MMP7
SCHEMBL9520501 0.79 ALDH1A1 (0.38) ALDH1A1MAPT
SCHEMBL7806807 0.78 USP2 (0.43) HTTPKMSMN1; SMN2MMP1MMP3
SCHEMBL31721849 0.75 POLB (0.43) SMN1; SMN2ITGB3ITGB1ITGAVITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed