SCHEMBL7806580

SCHEMBL7806580

Cc1[c]c(C)c(Cc2ccccc2)c(C)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 3/20 0.41
HPGD P15428 1/20 0.41
ENPP1 P22413 2/20 0.40
TLR8 Q9NR97 1/20 0.40
HTT P42858 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
POLB P06746 1/20 0.40
LMNA P02545 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
CYP2C9 P11712 2/20 0.38
FPR1 P21462 2/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10310928 0.72 TLR8 (0.61) ALDH1A1HSD17B10HPGDTLR8CYP2D6
SCHEMBL7819858 0.69 CALM1 (0.39) KDM4EALDH1A1HSD17B10HPGDPOLB
SCHEMBL19146528 0.68 CDC7 (0.43) KDM4EALDH1A1HSD17B10HPGDENPP1
SCHEMBL1900091 0.68 CYP2D6 (0.59) ALDH1A1TLR8CYP2D6
SCHEMBL28313729 0.67 CALM1 (0.58) KDM4EHTTSMN1; SMN2POLBLMNA
SCHEMBL11316141 0.67 LMNA (0.59) KDM4EALDH1A1HSD17B10SMN1; SMN2LMNA
Bicarbonate SCHEMBL11028140 0.67 ALDH1A1 (0.49) KDM4EALDH1A1HSD17B10HPGDTLR8
SCHEMBL9454757 0.66 SMN1; SMN2 (0.52) KDM4EALDH1A1HSD17B10HPGDHTT
SCHEMBL2820256 0.66 CALM1 (0.73) KDM4EALDH1A1HSD17B10HPGDCYP3A4
SCHEMBL5474691 0.66 OPRM1 (0.45) KDM4EALDH1A1HPGDSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091941-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2001-04-18 EP disclosed
US-6124463-A TREATMENT OF AFFECTIVE DISORDER, ANXIETY OR DEPRESSION DUPONT PHARMACEUTICALS (US) 2000-09-26 US disclosed
WO-2000001675-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 2000-01-13 WO disclosed