SCHEMBL7809185

SCHEMBL7809185

O=C1c2ccccc2C(=O)N1C[C@@H]1C[C@H](SC(c2ccccc2)(c2ccccc2)c2ccccc2)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
ATM Q13315 1/20 0.40
CCR5 P51681 3/20 0.38
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
ACHE P22303 1/20 0.35
AGTR1 P30556 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8781913 0.89 TDP1 (0.40) TDP1ATMCCR5ALDH1A1MAPT
SCHEMBL9363277 0.88 TDP1 (0.41) TDP1ATMCCR5ALDH1A1MAPT
SCHEMBL7805543 0.87 TDP1 (0.43) TDP1ATMCCR5ALDH1A1MAPT
SCHEMBL7806847 0.87 POLB (0.38) TDP1ALDH1A1
SCHEMBL9363174 0.87 CCR5 (0.42) TDP1ATMCCR5
SCHEMBL7805572 0.86 TDP1 (0.42) TDP1ATMCCR5ALDH1A1MAPT
SCHEMBL7811581 0.86 ATM (0.41) TDP1ATMCCR5ALDH1A1MAPT
SCHEMBL9138797 0.85 TDP1 (0.42) TDP1ATMCCR5ALDH1A1MAPT
SCHEMBL8781804 0.85 TDP1 (0.42) TDP1ATMCCR5ALDH1A1MAPT
SCHEMBL9363103 0.85 MGLL (0.41) TDP1ATMCCR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528678-B1 A pyrrolidylthiocarbapenem derivative with antibacterial activity SHIONOGI & CO (JP) 2001-05-23 EP disclosed
US-5703243-A Intermediates for pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1997-12-30 US disclosed
US-5317016-A Pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-05-31 US disclosed
EP-0528678-A1 A pyrrolidylthiocarbapenem derivative SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1993-02-24 EP disclosed