SCHEMBL7810348

SCHEMBL7810348

Cc1ccc(C(=S)c2ccc(F)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.62
NFE2L2 Q16236 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.44
CYP1A2 P05177 1/20 0.44
ALDH1A1 P00352 5/20 0.43
LMNA P02545 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 2/20 0.42
PAX8 Q06710 1/20 0.42
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 1/20 0.41
METTL3 Q86U44 1/20 0.40
HSD11B1 P28845 1/20 0.40
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4460667 0.87 ALDH1A1 (0.52) ACHESMN1; SMN2ALDH1A1LMNATDP1
SCHEMBL7810360 0.85 ACHE (0.42) ACHENFE2L2SMN1; SMN2CYP1A2ALDH1A1
SCHEMBL7810939 0.80 CTSL (0.56) ACHENFE2L2SMN1; SMN2ALDH1A1LMNA
Methyl Alcohol SCHEMBL27638432 0.79 ACHE (0.87) ACHENFE2L2SMN1; SMN2CYP1A2ALDH1A1
SCHEMBL7025938 0.79
SCHEMBL12689 0.79
SCHEMBL7802225 0.79 CES2 (0.47) ACHENFE2L2SMN1; SMN2ALDH1A1LMNA
SCHEMBL7814042 0.78 CES2 (0.46) ACHENFE2L2SMN1; SMN2ALDH1A1LMNA
SCHEMBL1127542 0.78 ALDH1A1 (0.44) ACHESMN1; SMN2ALDH1A1LMNATDP1
SCHEMBL6338854 0.78 CES2 (0.60) ACHESMN1; SMN2CYP1A2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843853-B Composition and method for manufacturing device using the same 东洋合成工业株式会社 2022-09-20 CN disclosed
EP-0891345-B1 NOVEL FURAN DIARYLMETHYLIDENE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THERAPEUTICAL USES THEREOF UNION PHARMA SCIENT APPL (FR) 2001-08-16 EP disclosed
US-6180651-B1 ANTIINFLAMMATORY AGENTS; ANALGESICS BRISTOL-MYERS SQUIBB 2001-01-30 US disclosed
WO-2000014082-A1 DIARYLMETHYLIDENE FURAN DERIVATIVES AS DRUGS WITH ANTI-INFLAMMATORY, ANALGESIC AND CHEMOPREVENTIVE PROPERTIES LABORATORIES UPSA (FR) 2000-03-16 WO disclosed
EP-0915850-A1 NOVEL CARBOCYCLIC DIARYLMETHYLENE DERIVATIVES, METHODS FOR PREPARING SAME, AND THERAPEUTICAL USES THEREOF LABORATOIRES UPSA (FR) 1999-05-19 EP disclosed
EP-0891345-A1 NOVEL FURAN DIARYLMETHYLIDENE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THERAPEUTICAL USES THEREOF LABORATOIRES UPSA (FR) 1999-01-20 EP disclosed
US-5840753-A ANTIINFLAMMATORY AGENTS, ANALGESICS LABORATORIES UPSA (FR) 1998-11-24 US disclosed
US-5807873-A Diarylmethylidenefuran derivatives and their uses in therapeutics LABORATORIES UPSA (FR) 1998-09-15 US disclosed
WO-1998005643-A1 NOVEL CARBOCYCLIC DIARYLMETHYLENE DERIVATIVES, METHODS FOR PREPARING SAME, AND THERAPEUTICAL USES THEREOF LABORATOIRES UPSA (FR) 1998-02-12 WO disclosed
US-5686460-A ANTIINFLAMMATORY AGENTS, ANALGESICS LABORATOIRES UPSA (FR) 1997-11-11 US disclosed
WO-1997037984-A1 NOVEL FURAN DIARYLMETHYLIDENE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THERAPEUTICAL USES THEREOF LABORATOIRES UPSA (FR) 1997-10-16 WO disclosed