SCHEMBL7811152

SCHEMBL7811152

O=c1[nH]c2cc(Cl)ccc2c(=O)cc1N1CCN(Cc2ccccc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.51
ALDH1A1 P00352 5/20 0.50
DRD4 P21917 3/20 0.49
DRD2 P14416 3/20 0.49
DRD3 P35462 2/20 0.49
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
CHRM1 P11229 1/20 0.47
HSD17B10 Q99714 2/20 0.47
TSHR P16473 2/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
TRPC5 Q9UL62 1/20 0.46
HTR1A P08908 1/20 0.46
SIGMAR1 Q99720 3/20 0.46
TRPV4 Q9HBA0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7802928 0.78 LMNA (0.45) ALDH1A1LMNAHPGDHSD17B10TSHR
SCHEMBL8173934 0.72 SIGMAR1 (0.70) ALDH1A1DRD4DRD2DRD3TSHR
Hydrochloric Acid SCHEMBL27955450 0.71 SIGMAR1 (0.61) ALDH1A1DRD4DRD2DRD3KDM4E
SCHEMBL8168486 0.71 SIGMAR1 (0.65) ALDH1A1DRD4DRD2DRD3SIGMAR1
SCHEMBL1783455 0.70 DRD4 (0.57) ALDH1A1DRD4DRD2DRD3LMNA
Hydrochloric Acid SCHEMBL11032993 0.70 DRD2 (0.57) ACHEALDH1A1DRD4DRD2DRD3
SCHEMBL7809286 0.70 LMNA (0.52) ALDH1A1LMNAHPGDHSD17B10KDM4E
SCHEMBL8311608 0.70 MAPT (0.62) ALDH1A1DRD4DRD2DRD3TRPC5
SCHEMBL11164060 0.69 DRD4 (0.55) ALDH1A1DRD4DRD2DRD3LMNA
SCHEMBL27470403 0.69 CYP3A4 (0.71) ALDH1A1DRD3CHRM1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0644878-B1 2,5-DIOXO-2,5-DIHYDRO-1H-BENZ b]AZEPINES AS NMDA RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2001-09-12 EP claimed
US-5492905-A NERVOUS SYSTEM DISORDERS ZENECA LIMITED (GB) 1996-02-20 US claimed