SCHEMBL7816337

SCHEMBL7816337

Cc1oc2c(NC(=O)c3c(Cl)cccc3Cl)cccc2c1COC(=O)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GHSR Q92847 2/20 0.41
GPR35 Q9HC97 3/20 0.40
MAPT P10636 8/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
POLB P06746 2/20 0.39
SLC16A3 O15427 1/20 0.39
TP53 P04637 2/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 2/20 0.38
CYP1A2 P05177 1/20 0.38
CRHBP P24387 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8804997 0.88 GPR35 (0.39) KDM4EALDH1A1NPSR1TSHRHSD17B10
SCHEMBL7823605 0.88 KMT2A (0.41) ALDH1A1GHSRMAPTMEN1KMT2A
SCHEMBL7832320 0.86 MAPT (0.42) ALDH1A1NPSR1TDP1GHSRGPR35
SCHEMBL8345228 0.85 PTGES (0.43) GHSRMAPTMEN1KMT2APOLB
SCHEMBL7827960 0.84 ALDH1A1 (0.40) ALDH1A1GHSRMAPTMEN1KMT2A
SCHEMBL7827815 0.84 MEN1 (0.44) ALDH1A1NPSR1GHSRGPR35MAPT
SCHEMBL7816960 0.83 KDM4E (0.38) KDM4ETDP1L3MBTL1GHSRGPR35
SCHEMBL7831438 0.82 AKR1B1 (0.42) HSD17B10GHSRGPR35MAPTMEN1
SCHEMBL7815783 0.82 MEN1 (0.44) ALDH1A1NPSR1GHSRGPR35MAPT
SCHEMBL7828350 0.82 TP53 (0.41) KDM4EALDH1A1TSHRTDP1GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757682-B1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO (JP) 2001-06-20 EP disclosed
US-5858995-A ADMINISTERING TO HUMANS AND ANIMALS IN THE TREATMENT OF DISEASES CAUSED BY ABNORMAL BONE METABOLISM FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-01-12 US disclosed
WO-1995029907-A1 BENZOFURAN DERIVATIVES USEFUL AS INHIBITORS OF BONE RESORPTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-11-09 WO disclosed