SCHEMBL7816658

SCHEMBL7816658

CCCCc1ccc2c(nc(CC)n2C)c1-c1cc(F)c(Cl)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
TLR7 Q9NYK1 2/20 0.30
AGTR1 P30556 1/20 0.30
AGTR2 P50052 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7813650 0.69 CYP11B2 (0.31)
SCHEMBL7814352 0.69 HCAR1 (0.34)
SCHEMBL11923731 0.62 DPP4 (0.41)
SCHEMBL12263310 0.62 MEN1 (0.43)
SCHEMBL28230824 0.62 TLR8 (0.43) TLR7
SCHEMBL7817046 0.62 POLB (0.33)
SCHEMBL7813559 0.59 TLR8 (0.41)
SCHEMBL24401836 0.58 KDM4E (0.32) TLR7
SCHEMBL12362580 0.58 HSP90AB1 (0.49) TLR7
SCHEMBL29924487 0.57 TYR (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091941-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2001-04-18 EP claimed
WO-2000001675-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 2000-01-13 WO claimed