SCHEMBL7814352

SCHEMBL7814352

CCCc1ccc2c(nc(CC)n2-c2ccccc2)c1-c1cc(Cl)c(Cl)cc1Cl

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.34
PDE10A Q9Y233 9/20 0.33
CYP1A2 P05177 2/20 0.33
MAT2A P31153 1/20 0.33
PI4KA P42356 1/20 0.32
PI4K2B Q8TCG2 1/20 0.32
PI4K2A Q9BTU6 1/20 0.32
PI4KB Q9UBF8 1/20 0.32
DCTPP1 Q9H773 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
PPARG P37231 1/20 0.32
P2RX7 Q99572 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7813650 0.78 CYP11B2 (0.31)
SCHEMBL7817046 0.71 POLB (0.33) CYP1A2ALDH1A1
SCHEMBL6447298 0.69 DCTPP1 (0.49) PDE10ACYP1A2MAT2ADCTPP1ALDH1A1
SCHEMBL10815729 0.66 PPARG (0.47) HCAR1PDE10ACYP1A2PI4KAPI4K2B
SCHEMBL10818689 0.63 CYP1A2 (0.54) PDE10ACYP1A2MAT2ASMN1; SMN2
SCHEMBL23105555 0.63 L3MBTL1 (0.45) PDE10ACYP1A2SMN1; SMN2NR1H2NR1H3
SCHEMBL25112562 0.63 PDE10A (0.63) PDE10AALDH1A1
SCHEMBL10817241 0.62 PPARG (0.48) HCAR1PDE10ACYP1A2PI4KAPI4K2B
SCHEMBL10817583 0.61 PDE10A (0.56) HCAR1PDE10ACYP1A2MAT2APPARG
SCHEMBL1623493 0.61 PPARG (0.39) NR1H2NR1H3PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091941-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2001-04-18 EP claimed
WO-2000001675-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 2000-01-13 WO claimed
EP-1091941-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2001-04-18 EP disclosed
WO-2000001675-A1 NOVEL BENZIMIDAZOLES AS CORTICOTROPIN RELEASE FACTOR ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 2000-01-13 WO disclosed