SCHEMBL7818154

SCHEMBL7818154

O=C(NCCNc1cc(=O)c2ccccc2[nH]1)c1cnc(Cl)c(Cl)c1

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
MARS1 P56192 1/20 0.46
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7815904 0.94 MARS1 (0.52) MARS1
SCHEMBL7821468 0.78 MARS1 (0.60) ALDH1A1MARS1
SCHEMBL7818445 0.78 KDM4E (0.46) ALDH1A1MARS1KMT2A
SCHEMBL7818007 0.70 MARS1 (0.48) ALDH1A1MARS1
SCHEMBL5668076 0.69 MARS1 (0.59) MARS1
SCHEMBL7488352 0.69 ALDH1A1 (0.54) ALDH1A1OPRM1OPRD1KMT2A
Ammonia Solution, Strong SCHEMBL5667906 0.68 MARS1 (0.58) MARS1
Hydrochloric Acid SCHEMBL5669755 0.68 MARS1 (0.58) MARS1
Hydrochloric Acid SCHEMBL7995914 0.68 MARS1 (0.54) MARS1
Hydrochloric Acid SCHEMBL7992242 0.67 MARS1 (0.57) MARS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6320051-B1 AMINO(NH) OR OXYGEN(O) SUBSTITUTED, ENZYME INHIBITORS OF STAPHLOCCOCUS AUREUS METHIONYL T-RNA SYNTHETASE (MRS); ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2001-11-20 US claimed
EP-1084110-A1 QUINOLONES USED AS MRS INHIBITORS AND BACTERICIDES SMITHKLINE BEECHAM PLC (GB) 2001-03-21 EP claimed
WO-1999055677-A1 QUINOLONES USED AS MRS INHIBITORS AND BACTERICIDES SMITHKLINE BEECHAM PLC (GB) 1999-11-04 WO claimed
US-6320051-B1 AMINO(NH) OR OXYGEN(O) SUBSTITUTED, ENZYME INHIBITORS OF STAPHLOCCOCUS AUREUS METHIONYL T-RNA SYNTHETASE (MRS); ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2001-11-20 US disclosed