SCHEMBL7819686

SCHEMBL7819686

O=C1c2cc[n+]([O-])cc2C(=O)c2c(Cl)ccc(F)c21

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.38
GPR84 Q9NQS5 2/20 0.33
CCR9 P51686 5/20 0.32
PTGS2 P35354 6/20 0.31
PTGS1 P23219 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546620 0.91 MEN1 (0.32) GPR84
SCHEMBL7817749 0.72 LMNA (0.37) PTGS2PTGS1
SCHEMBL7825262 0.72 KMT2A (0.39) CCR9
SCHEMBL7818383 0.72 LMNA (0.37) PTGS2PTGS1
SCHEMBL7830253 0.69 MEN1 (0.52)
SCHEMBL7806728 0.69 CDC25B (0.56) ADORA2APTGS2PTGS1
SCHEMBL29780065 0.66 GPR84 (0.40) GPR84
SCHEMBL6674009 0.65 CSNK2A2 (0.44) ADORA2A
SCHEMBL8540388 0.65 ECE1 (0.45) CCR9PTGS2
SCHEMBL308115 0.64 ADORA2A (0.76) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
EP-0750619-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-02 EP disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed