SCHEMBL7820192

SCHEMBL7820192

O=C(O)c1cc(Br)ccc1NS(=O)(=O)c1cccc2nsnc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 1.00
METAP2 P50579 1/20 1.00
KMT2A Q03164 1/20 1.00
L3MBTL1 Q9Y468 2/20 0.73
ATM Q13315 1/20 0.73
CCKBR P32239 10/20 0.72
POLB P06746 2/20 0.67
CCKAR P32238 4/20 0.63
CTDSP1 Q9GZU7 2/20 0.62
GAA P10253 1/20 0.58
MAPT P10636 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
DUSP3 P51452 1/20 0.56
PTPN5 P54829 1/20 0.56
CASP6 P55212 1/20 0.56
PTPN11 Q06124 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3741036 0.91 MEN1 (0.84) MEN1METAP2KMT2AL3MBTL1ATM
SCHEMBL3745368 0.87 MEN1 (0.77) MEN1METAP2KMT2AL3MBTL1ATM
SCHEMBL7213043 0.86 MEN1 (0.76) MEN1METAP2KMT2AL3MBTL1ATM
SCHEMBL3899468 0.85 L3MBTL1 (1.00) MEN1METAP2KMT2AL3MBTL1ATM
SCHEMBL13792850 0.84 CCKBR (1.00) MEN1METAP2KMT2ACCKBR
SCHEMBL3900101 0.83 L3MBTL1 (0.75) MEN1METAP2KMT2AL3MBTL1ATM
SCHEMBL3749920 0.83 POLB (0.72) MEN1METAP2KMT2AL3MBTL1ATM
SCHEMBL3745619 0.82 MEN1 (0.69) MEN1METAP2KMT2AL3MBTL1ATM
SCHEMBL21857833 0.81 L3MBTL1 (0.82) MEN1METAP2KMT2AL3MBTL1ATM
SCHEMBL3746034 0.80 CCKBR (0.74) L3MBTL1ATMCCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120010290-A1 Methods of Treating an Overweight or Obese Subject ZAFGEN, INC. 2012-01-12 US disclosed
US-20120010290-A1 Methods of Treating an Overweight or Obese Subject ZAFGEN, INC. 2012-01-12 US disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010290-A1 Methods of Treating an Overweight or Obese Subject METAP2, METAP1, ACER2 MEN1 1391/4885METAP2 1/4885KMT2A 380/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.