SCHEMBL7822244

SCHEMBL7822244

Cc1c([N+](=O)[O-])c(=O)oc2c(C)c3c(cc12)CC(CBr)O3

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 2/20 0.32
TSHR P16473 2/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
MAPT P10636 4/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 2/20 0.31
HSD17B10 Q99714 1/20 0.31
GPR35 Q9HC97 1/20 0.31
LMNA P02545 1/20 0.30
KDM4E B2RXH2 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10379963 0.83 MAPT (0.38) MCL1TSHRMAPK1HTTMAPT
SCHEMBL7814957 0.82 HSD17B3 (0.34) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7829873 0.80 HSD17B3 (0.38) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7483011 0.78 MAOA (0.43) MCL1TSHRMAPK1HTTMAPT
SCHEMBL7822820 0.73 ALDH1A1 (0.42) TSHRMAPK1HTTMAPTSMN1; SMN2
SCHEMBL7822480 0.71 TSHR (0.34) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7823020 0.71 HSD17B3 (0.34) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7822789 0.68 HSD17B3 (0.38) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7822838 0.68 KDM4E (0.39) MAPK1HTTMAPTSMN1; SMN2ALDH1A1
SCHEMBL7814575 0.68 KMT2A (0.38) TSHRMAPK1HTTMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133498-A2 AMINO-AND MERCURIO-SUBSTITUTED 4', 5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2001-09-19 EP claimed
WO-2000031081-A2 AMINO- AND MERCURIO-SUBSTITUTED 4',5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2000-06-02 WO claimed
EP-1133498-A2 AMINO-AND MERCURIO-SUBSTITUTED 4', 5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2001-09-19 EP disclosed
US-6255324-B1 MICROBIOCIDES; SKIN DISORDERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2001-07-03 US disclosed
WO-2000031081-A2 AMINO- AND MERCURIO-SUBSTITUTED 4',5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2000-06-02 WO disclosed