SCHEMBL7822480

SCHEMBL7822480

Cc1c(I)c(=O)oc2c(C)c3c(cc12)CC(CI)O3

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.34
MAPK1 P28482 2/20 0.34
HTT P42858 1/20 0.34
MAPT P10636 4/20 0.33
ALDH1A1 P00352 3/20 0.33
HSD17B10 Q99714 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CNR2 P34972 3/20 0.32
GPR55 Q9Y2T6 3/20 0.32
CNR1 P21554 1/20 0.32
NQO1 P15559 1/20 0.32
HPGD P15428 1/20 0.30
TP53 P04637 2/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7823020 0.86 HSD17B3 (0.34) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7822820 0.86 ALDH1A1 (0.42) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7822789 0.83 HSD17B3 (0.38) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7824606 0.83 MAPT (0.31) TSHRMAPK1HTTMAPTTP53
SCHEMBL7822499 0.82 MAOA (0.43) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7814954 0.75 ALDH1A1 (0.43) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7814957 0.74 HSD17B3 (0.34) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7484595 0.72 TSHR (0.32) TSHRMAPK1HTTALDH1A1HSD17B10
SCHEMBL7829873 0.71 HSD17B3 (0.38) TSHRMAPK1HTTMAPTALDH1A1
SCHEMBL7822244 0.71 MCL1 (0.32) TSHRMAPK1HTTMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133498-A2 AMINO-AND MERCURIO-SUBSTITUTED 4', 5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2001-09-19 EP claimed
WO-2000031081-A2 AMINO- AND MERCURIO-SUBSTITUTED 4',5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2000-06-02 WO claimed
EP-1133498-A2 AMINO-AND MERCURIO-SUBSTITUTED 4', 5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2001-09-19 EP disclosed
US-6255324-B1 MICROBIOCIDES; SKIN DISORDERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2001-07-03 US disclosed
WO-2000031081-A2 AMINO- AND MERCURIO-SUBSTITUTED 4',5'-DIHYDROPSORALENS AND THERAPEUTICAL USES THEREOF BUCKMAN LABORATORIES INTERNATIONAL, INC. (US) 2000-06-02 WO disclosed