SCHEMBL7822307

SCHEMBL7822307

COc1ccc(/C=N/c2ccc(O[Si](C)(C)C(C)(C)C)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100B P04271 1/20 0.59
PTGS2 P35354 3/20 0.52
CA2 P00918 2/20 0.52
PTGS1 P23219 1/20 0.52
CA12 O43570 1/20 0.52
CA9 Q16790 1/20 0.52
ACHE P22303 2/20 0.46
ALDH1A1 P00352 4/20 0.44
GAA P10253 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.42
CA1 P00915 1/20 0.41
APP P05067 1/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7822309 1.00 S100B (0.59) S100BPTGS2CA2PTGS1CA12
SCHEMBL3498339 0.87 S100B (0.43) S100BPTGS2CA2PTGS1CA12
SCHEMBL2746628 0.87 CA2 (0.44) S100BPTGS2CA2PTGS1CA12
SCHEMBL3499959 0.87 S100B (0.43) S100BPTGS2CA2PTGS1CA12
SCHEMBL2746630 0.87 CA2 (0.44) S100BPTGS2CA2PTGS1CA12
SCHEMBL12416630 0.82 S100B (0.82) S100BPTGS2CA2PTGS1CA12
SCHEMBL10733277 0.82 S100B (0.82) S100BPTGS2CA2PTGS1CA12
SCHEMBL10412841 0.82 S100B (0.82) S100BPTGS2CA2PTGS1CA12
SCHEMBL10733285 0.82 S100B (0.82) S100BPTGS2CA2PTGS1CA12
SCHEMBL2010515 0.82 S100B (0.82) S100BPTGS2CA2PTGS1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0681569-B1 SPIROCYCLOALKYL-SUBSTITUTED AZETIDINONES USEFUL AS HYPOCHOLESTEROLEMIC AGENTS SCHERING CORP (US) 2001-03-21 EP disclosed
US-5698548-A Spirocycloalkyl-substituted azetidinones useful as hypocholesterolemic agents SCHERING CORPORATION (US) 1997-12-16 US disclosed