SCHEMBL7822347

SCHEMBL7822347

O=C(Cc1nc2cc(-n3ccnc3)ccc2[nH]1)Nc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
PORCN Q9H237 2/20 0.50
MEN1 O00255 1/20 0.50
POLB P06746 1/20 0.50
KMT2A Q03164 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 1/20 0.48
F9 P00740 1/20 0.45
PARP1 P09874 1/20 0.45
PARP3 Q9Y6F1 1/20 0.45
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
WNT3A P56704 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB3 P13945 1/20 0.43
ACP1 P24666 1/20 0.42
LMNA P02545 2/20 0.42
MAPK1 P28482 1/20 0.42
PIK3CD O00329 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7822350 0.92 ALDH1A1 (0.50) ALDH1A1PORCNMEN1POLBKMT2A
SCHEMBL7822768 0.82 IDH1 (0.48) ALDH1A1PORCNMEN1KMT2ACYP3A4
SCHEMBL7836354 0.80 CYP4Z1 (0.55) ALDH1A1POLBKMT2AF9SMN1; SMN2
SCHEMBL7835277 0.80 F9 (0.41) PORCNMEN1KMT2ACYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8148418 0.79 CYP4Z1 (0.54) ALDH1A1POLBKMT2AF9SMN1; SMN2
SCHEMBL4071088 0.77 HSD17B10 (0.56) ALDH1A1MEN1KMT2ACYP3A4CYP2D6
SCHEMBL7407358 0.77 CBFB (0.50) POLBF9RAB9ALMNACYP19A1
SCHEMBL7822232 0.77 TNIK (0.45) ALDH1A1PORCNMEN1POLBKMT2A
Hydrochloric Acid SCHEMBL8155236 0.77 F9 (0.46) TDP1F9LMNACYP19A1CYP11B1
SCHEMBL15685943 0.76 ALDH1A1 (0.74) ALDH1A1MEN1POLBKMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed