SCHEMBL7822667

SCHEMBL7822667

N#Cc1c(-c2c[nH]c3ccccc23)[nH]c(=O)n1-c1cccc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.41
MET P08581 2/20 0.41
EGFR P00533 1/20 0.41
BRAF P15056 1/20 0.41
CDK6 Q00534 1/20 0.41
SIRT2 Q8IXJ6 3/20 0.38
SIRT1 Q96EB6 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PRKCB P05771 2/20 0.37
PRKCA P17252 2/20 0.37
PRKD3 O94806 1/20 0.37
CCNB2 O95067 1/20 0.37
CCNE2 O96020 1/20 0.37
ABL1 P00519 1/20 0.37
PRKCG P05129 1/20 0.37
CDK1 P06493 1/20 0.37
PIM1 P11309 1/20 0.37
CCNB1 P14635 1/20 0.37
PRKACA P17612 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976408 0.82 MEN1 (0.40) CDK4METEGFRBRAFCDK6
SCHEMBL7004515 0.77 SIRT2 (0.43) CDK4SIRT2SIRT1MEN1KMT2A
SCHEMBL7820421 0.72 PDE9A (0.40) CDK4METEGFRBRAFCDK6
SCHEMBL6589577 0.71 MAPK1 (0.45) CDK4CDK6SIRT2SIRT1MEN1
Acetic Acid SCHEMBL7840658 0.69 NPEPPS (0.33) CAMK2DITGA4ITGB7
SCHEMBL7819614 0.68 MPO (0.36) CDK4METEGFRBRAFCDK6
SCHEMBL6976268 0.68 NPEPPS (0.63) GAAHCAR1
SCHEMBL7821934 0.66 PDE9A (0.33) CDK4METEGFRBRAFCDK6
SCHEMBL7010190 0.65 NT5E (0.45) CDK4SIRT2SIRT1MEN1KMT2A
SCHEMBL29326335 0.65 NPEPPS (0.43) PIM1GAAMCL1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095039-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS AstraZeneca AB (SE) 2001-05-02 EP disclosed
WO-2000002877-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2000-01-20 WO disclosed