SCHEMBL7819614

SCHEMBL7819614

N#Cc1c(-c2c(CCN)[nH]c3ccccc23)[nH]c(=O)n1-c1c[nH]c2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2A6 P11509 1/20 0.36
NFKB1 P19838 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR7 P34969 1/20 0.36
CTSK P43235 1/20 0.36
HTR6 P50406 1/20 0.36
CYP2A13 Q16696 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
PMP22 Q01453 1/20 0.36
PDE9A O76083 5/20 0.35
PDE1C Q14123 1/20 0.35
IMPDH2 P12268 1/20 0.33
IMPDH1 P20839 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7821934 0.93 PDE9A (0.33) MPOCYP1A2CYP3A4CYP2D6CYP2A6
SCHEMBL7823271 0.88 ALDH1A1 (0.35) PDE9APDE1CIMPDH2IMPDH1CAMK2D
Trifluoroacetic Acid SCHEMBL7838986 0.86 SSTR4 (0.33) PDE9A
SCHEMBL7819396 0.86 IDO1 (0.33) CYP3A4PDE9ARPS6KB1STAT3
SCHEMBL7826355 0.85 ALDH1A1 (0.32) PDE9ASTAT3
SCHEMBL7812318 0.84 PRKCB (0.33) PDE9ANPEPPSEGFRMETCDK4
SCHEMBL7826816 0.84 ALDH1A1 (0.33) PDE9ASTAT3
SCHEMBL7820421 0.82 PDE9A (0.40) HTR2AHTR2CHTR6PDE9APDE1C
Trifluoroacetic Acid SCHEMBL7839584 0.80 OXER1 (0.30)
Trifluoroacetic Acid SCHEMBL7828206 0.78 TPSAB1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1095039-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS AstraZeneca AB (SE) 2001-05-02 EP claimed
WO-2000002877-A2 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2000-01-20 WO claimed