SCHEMBL7823002

SCHEMBL7823002

NC(=O)Nc1ccc(Oc2ccc(O)cc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PEPD P12955 1/20 0.77
HSD17B10 Q99714 1/20 0.62
PARP10 Q53GL7 1/20 0.58
ALDH1A1 P00352 5/20 0.56
GLA P06280 2/20 0.56
CYP3A4 P08684 2/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
HPGD P15428 1/20 0.55
ALOX12 P18054 1/20 0.55
CYP2C19 P33261 1/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
ESR1 P03372 1/20 0.54
ESR2 Q92731 1/20 0.54
GAA P10253 3/20 0.53
MAPT P10636 3/20 0.53
GFER P55789 2/20 0.53
KDM4E B2RXH2 1/20 0.53
THRB P10828 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1322717 0.88 PEPD (1.00) PEPDALDH1A1GLACYP3A4MEN1
SCHEMBL5528916 0.85 SMN1; SMN2 (0.66) HSD17B10PARP10ALDH1A1HPGDGAA
SCHEMBL17628546 0.84 MAOA (0.64) PEPDMEN1KMT2AESR1ESR2
SCHEMBL4092732 0.83 NPC1 (0.78) PEPDHSD17B10ALDH1A1GLACYP3A4
SCHEMBL13750226 0.83 KIF11 (0.70) PEPDHSD17B10ALDH1A1GLACYP3A4
SCHEMBL5008975 0.81 HSD17B10 (0.58) PEPDHSD17B10ALDH1A1GLACYP3A4
SCHEMBL2844063 0.81 KMT2A (0.77) ALDH1A1CYP3A4HPGDMEN1KMT2A
SCHEMBL5062623 0.78 PEPD (0.80) PEPDHSD17B10ALDH1A1GLAMEN1
SCHEMBL11831801 0.78 MEN1 (0.77) HSD17B10ALDH1A1MEN1KMT2AGAA
SCHEMBL21550458 0.77 PEPD (0.77) PEPDALDH1A1GLACYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047418-A4 INHIBITION OF RAF KINASE USING SUBSTITUTED HETEROCYCLIC UREAS BAYER AG (US) 2001-02-07 EP claimed
EP-1047418-A1 INHIBITION OF RAF KINASE USING SUBSTITUTED HETEROCYCLIC UREAS Bayer Corporation (US) 2000-11-02 EP claimed
WO-1999032106-A1 INHIBITION OF RAF KINASE USING SUBSTITUTED HETEROCYCLIC UREAS BAYER CORPORATION (US) 1999-07-01 WO claimed