SCHEMBL7823286

SCHEMBL7823286

OCCCc1nc2cccnc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.46
POLB P06746 1/20 0.45
PKM P14618 1/20 0.42
RIPK1 Q13546 2/20 0.40
EGFR P00533 2/20 0.39
MAPK14 Q16539 2/20 0.39
PARP1 P09874 1/20 0.37
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7026169 0.84 PARP1 (0.54) POLBPARP1NPC1
SCHEMBL4347806 0.83 RIPK1 (0.43) RIPK1NPC1LMNARAB9A
SCHEMBL9853629 0.80 KDM4C (0.48) POLBPARP1NPC1LMNARAB9A
SCHEMBL7002587 0.79 GAA (0.42) POLBPKMEGFRNPC1LMNA
SCHEMBL30831392 0.78 POLB (0.43) POLBPKMLMNAHCAR2
SCHEMBL31660973 0.76 CYP1A2 (0.37) POLBPARP1NPC1LMNARAB9A
SCHEMBL13233304 0.76 CYP1A2 (0.43) POLBNPC1LMNARAB9A
SCHEMBL4361327 0.76 DDAH1 (0.55) POLBPKMNPC1LMNARAB9A
SCHEMBL18291869 0.76 ALDH1A1 (0.38) POLBPKMRIPK1PARP1NPC1
SCHEMBL5264712 0.76 ALDH1A1 (0.38) POLBPKMPARP1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676398-B1 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO CO (JP) 2001-10-24 EP disclosed
US-6117893-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 2000-09-12 US disclosed
EP-1022274-A1 Oxazolidinedione and Thiazolidinedione derivatves, their preparation and their use Sankyo Company Limited (JP) 2000-07-26 EP disclosed
US-5977365-A HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
US-5962470-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 1999-10-05 US disclosed
US-5834501-A TREATING DIABETES OR HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 1998-11-10 US disclosed
US-5739345-A HYPOGLYCEMIC AND ANTIDIABETIC AGENTS SANKYO COMPANY, LIMITED (JP) 1998-04-14 US disclosed
US-5624935-A ANTIDIABETIC AGENTS, HYPOGLYCEMIC AGENTS OR ANTILIPEMIC AGENTS SANKYO COMPANY, LIMITED 1997-04-29 US disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed