SCHEMBL7823372

SCHEMBL7823372

COc1cccc2c1C(C)(C)C(=O)N2CCO

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA1A P35348 1/20 0.41
ALDH1A1 P00352 2/20 0.39
AADAT Q8N5Z0 1/20 0.38
SCN9A Q15858 1/20 0.38
TP53 P04637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
MGLL Q99685 1/20 0.36
ALOX15 P16050 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833326 0.81 TP53 (0.41) CYP3A4TSHRTP53KDM4EMAPT
SCHEMBL3483987 0.79 MGLL (0.42) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL7014237 0.74 TP53 (0.52) CYP1A2CYP3A4ALDH1A1TP53MEN1
SCHEMBL31559833 0.74 TP53 (0.52) CYP1A2CYP3A4ALDH1A1TP53MEN1
SCHEMBL7062684 0.72 CYP2D6 (0.73) CYP3A4MEN1MAPK1KMT2ADRD2
SCHEMBL7825844 0.67 PARK7 (0.47) CYP3A4MEN1MAPTMAPK1KMT2A
SCHEMBL5007556 0.67 HSPA9 (0.39) CYP3A4TP53KDM4EMEN1MAPT
SCHEMBL7837760 0.66 TP53 (0.44) CYP3A4TSHRTP53KDM4EMEN1
SCHEMBL30972520 0.66 ALDH1A1 (0.43) TSHRALDH1A1AADATTP53KDM4E
SCHEMBL28850390 0.65 ALDH1A1 (0.54) CYP1A2CYP3A4ALDH1A1SCN9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780388-B1 5HT1Dalpha and 5HT2A ligands LILLY CO ELI (GB) 2001-08-16 EP disclosed
US-5773448-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY LIMITED (GB) 1998-06-30 US disclosed
EP-0780388-A1 5HT1Dalpha and 5HT2A ligands LILLY INDUSTRIES LIMITED (GB) 1997-06-25 EP disclosed