SCHEMBL7823403

SCHEMBL7823403

O=C(O)c1cnncc1C(=O)c1cc(F)ccc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.52
CES1 P23141 3/20 0.52
KEAP1 Q14145 2/20 0.47
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
MEN1 O00255 2/20 0.39
HPGD P15428 2/20 0.39
KMT2A Q03164 2/20 0.39
TTR P02766 2/20 0.39
USP2 O75604 1/20 0.39
DHFR P00374 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
LMNA P02545 1/20 0.39
ALB P02768 1/20 0.39
HMGB1 P09429 1/20 0.39
CXCL12 P48061 1/20 0.39
HIF1A Q16665 1/20 0.39
SLC22A6 Q4U2R8 1/20 0.39
ACMSD Q8TDX5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7772555 0.83 CES2 (0.47) CES2CES1KEAP1ALDH1A1KDM4E
SCHEMBL7766931 0.83 CES2 (0.47) CES2CES1KEAP1ALDH1A1KDM4E
SCHEMBL27673772 0.82 CES2 (0.74) CES2CES1KEAP1ALDH1A1MEN1
SCHEMBL115334 0.80 CES2 (0.71) CES2CES1KEAP1ALDH1A1KDM4E
SCHEMBL28742361 0.78 CES2 (0.68) CES2CES1KEAP1ALDH1A1KDM4E
SCHEMBL29798953 0.78 CES2 (0.68) CES2CES1KEAP1ALDH1A1KDM4E
SCHEMBL7818617 0.72 CES2 (0.50) CES2CES1KEAP1ALDH1A1KDM4E
SCHEMBL8545735 0.72 KDM4E (0.56) CES2CES1KEAP1ALDH1A1KDM4E
SCHEMBL8542675 0.72 KDM4E (0.56) CES2CES1KEAP1ALDH1A1KDM4E
SCHEMBL29367263 0.72 CES2 (0.59) CES2CES1KEAP1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
EP-0750619-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-02 EP disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed