SCHEMBL7823957

SCHEMBL7823957

COc1ccc2c(c1)CC1(CC2)COCC(=O)N1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.54
BACE1 P56817 2/20 0.40
PRNP P04156 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
OTUD7B Q6GQQ9 1/20 0.37
PDE7A Q13946 2/20 0.36
AR P10275 2/20 0.36
METAP1 P53582 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7828016 0.95 ADRA2A (0.54) ADRA2ABACE1PRNPSMN1; SMN2PDE3B
SCHEMBL7815545 0.83 ALDH1A1 (0.40) ADRA2ASMN1; SMN2
SCHEMBL743822 0.80 ADRA2A (0.43) ADRA2ABACE1PRNPSMN1; SMN2PDE3B
SCHEMBL9047053 0.79 ADRA2A (0.55) ADRA2APRNPSMN1; SMN2
SCHEMBL7824594 0.78 ADRA2A (0.45) ADRA2ASMN1; SMN2
Hydrochloric Acid SCHEMBL7830547 0.78 ADRA2A (0.54) ADRA2ASMN1; SMN2
SCHEMBL9049906 0.73 ADRA2A (0.55) ADRA2APRNPSMN1; SMN2
Hydrochloric Acid SCHEMBL7826706 0.72 ADRA2A (0.54) ADRA2ASMN1; SMN2
Hydrochloric Acid SCHEMBL29051753 0.69 ADRA2A (0.56) ADRA2APRNP
Hydrochloric Acid SCHEMBL30468426 0.69 ADRA2A (0.56) ADRA2APRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712845-B1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-17 EP disclosed
US-5633248-A GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS, DIARYLALKYLIDENEDIAMINES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-27 US disclosed
US-5591849-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, INHIBITORS OF AMINE, AMINE OXIDASE B, AND CALCIUM ION UPTAKE, NEUROPATHY, DYSMNESIA TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-07 US disclosed
EP-0712845-A1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-22 EP disclosed
EP-0670313-A1 Spiro compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-09-06 EP disclosed