SCHEMBL7815545

SCHEMBL7815545

COc1cc2c(cc1OC)CC1(CC2)COCC(=O)N1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
RAB9A P51151 1/20 0.40
MAPK1 P28482 1/20 0.37
CYP3A4 P08684 1/20 0.37
KDM4E B2RXH2 2/20 0.35
CHRNA7 P36544 2/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ADRA2A P08913 2/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
ABCB1 P08183 1/20 0.33
TSHR P16473 1/20 0.33
MAOA P21397 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7828016 0.83 ADRA2A (0.54) CHRNA7SMN1; SMN2ADRA2A
SCHEMBL7823957 0.83 ADRA2A (0.54) SMN1; SMN2ADRA2A
SCHEMBL9052613 0.77 ALDH1A1 (0.38) ALDH1A1RAB9ACYP3A4KDM4ECHRNA7
Hydrochloric Acid SCHEMBL7828652 0.76 ALDH1A1 (0.37) ALDH1A1RAB9ACYP3A4KDM4ECHRNA7
SCHEMBL7824594 0.76 ADRA2A (0.45) ALDH1A1SMN1; SMN2ADRA2ATSHR
SCHEMBL11073395 0.73 GAA (0.39) ALDH1A1RAB9AMAPK1CYP3A4KDM4E
SCHEMBL18630670 0.68
Hydrochloric Acid SCHEMBL7815957 0.68 ALDH1A1 (0.49) ALDH1A1RAB9AMAPK1CYP3A4KDM4E
SCHEMBL7822652 0.67 ACHE (0.41) ALDH1A1RAB9AMAPK1KDM4ECHRNA7
SCHEMBL7827339 0.66 GAA (0.42) ALDH1A1GAASMN1; SMN2ABCB1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712845-B1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-17 EP disclosed
US-5633248-A GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS, DIARYLALKYLIDENEDIAMINES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-27 US disclosed
US-5591849-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, INHIBITORS OF AMINE, AMINE OXIDASE B, AND CALCIUM ION UPTAKE, NEUROPATHY, DYSMNESIA TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-07 US disclosed
EP-0712845-A1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-22 EP disclosed
EP-0670313-A1 Spiro compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-09-06 EP disclosed