SCHEMBL7824635

SCHEMBL7824635

O=CNc1sccc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN2 P17706 1/20 0.58
PTPRB P23467 1/20 0.58
PTPN6 P29350 1/20 0.58
ABCC1 P33527 2/20 0.46
ACLY P53396 1/20 0.45
HCAR2 Q8TDS4 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
NR4A1 P22736 1/20 0.41
RECQL P46063 1/20 0.41
ESR2 Q92731 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL546304 0.83 PTK2 (0.59) ALDH1A1MAPK1MEN1KMT2AMAPT
SCHEMBL13764835 0.76 PTPN2 (0.72) PTPN2PTPRBPTPN6ABCC1ACLY
SCHEMBL3576557 0.76 PTPN2 (0.61) PTPN2PTPRBPTPN6ABCC1ACLY
SCHEMBL12756123 0.76 PTPN2 (0.61) PTPN2PTPRBPTPN6ABCC1ACLY
SCHEMBL6643211 0.75 ALDH1A1 (0.53) KDM4EALDH1A1GAAHPGDMEN1
SCHEMBL5836577 0.73 PTPN2 (1.00) PTPN2PTPRBPTPN6ABCC1ACLY
SCHEMBL5550829 0.73 PTPN2 (0.68) PTPN2PTPRBPTPN6ABCC1HCAR2
SCHEMBL1704195 0.73 PTK2 (0.71) PTPN2PTPRBPTPN6ABCC1ACLY
SCHEMBL1992502 0.73 CYP3A4 (0.51) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL10743903 0.72 PTPN2 (0.44) PTPN2PTPRBPTPN6ABCC1ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346861-B1 THIOPHENE CONTAINING ANALOGUES OF FLUCONAZOLE AS ANTIFUNGAL AGENTS AND PROCESS THEREOF COUNCIL SCIENT IND RES (IN) 2013-01-23 EP claimed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed
US-4658040-A Process for manufacturing heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-04-14 US disclosed
US-4108867-A 2-Aminothiophenes IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1978-08-22 US disclosed