SCHEMBL7824847

SCHEMBL7824847

CCOC(=O)Cc1cccc2c1CC(n1cc(CP(=O)(O)O)nc1C(=O)OCC)C2=O

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.33
P2RX7 Q99572 1/20 0.33
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
HSD17B10 Q99714 1/20 0.32
FGFR1 P11362 1/20 0.31
FLT1 P17948 1/20 0.31
FGFR3 P22607 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8020015 0.92 P2RX7 (0.33) ALDH1A1GAAP2RX7MAPTHTT
SCHEMBL8013600 0.91 ALDH1A1 (0.36) ALDH1A1GAAP2RX7MAPTHTT
SCHEMBL7845523 0.88 ALDH1A1 (0.34) ALDH1A1GAAP2RX7MAPTHTT
SCHEMBL8099222 0.86 GAA (0.38) ALDH1A1GAAP2RX7MAPTHTT
SCHEMBL8090703 0.85 GAA (0.33) ALDH1A1GAAP2RX7MAPTHTT
SCHEMBL7819659 0.84 ALDH1A1 (0.36) ALDH1A1GAAP2RX7MAPTHTT
SCHEMBL8593496 0.83 ALDH1A1 (0.34) ALDH1A1GAAP2RX7MAPTHTT
SCHEMBL8012714 0.82 GAA (0.36) ALDH1A1GAAP2RX7MAPTHSD17B10
SCHEMBL8017443 0.82 FGFR1 (0.31) ALDH1A1GAAFGFR1FLT1FGFR3
SCHEMBL8015909 0.81 PARP1 (0.36) ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880522-B1 5H,10H-IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZINE-4-ONE DERIVATIVES AMPA AND NMDA RECEPTORS ANTAGONISTS, PREPARATION THEREOF, INTERMEDIATES THEREOF AND DRUGS CONTAINING SAME AVENTIS PHARMA SA (FR) 2001-09-19 EP disclosed
EP-0880522-A1 5H,10H-IMIDAZO 1,2-a]INDENO 1,2-e]PYRAZINE-4-ONE DERIVATIVES, PREPARATION THEREOF, INTERMEDIATES THEREOF AND DRUGS CONTAINING SAME Aventis Pharma S.A. (FR) 1998-12-02 EP disclosed
WO-1997025328-A1 5H,10H-IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZINE-4-ONE DERIVATIVES, PREPARATION THEREOF, INTERMEDIATES THEREOF AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1997-07-17 WO disclosed