SCHEMBL7828548

SCHEMBL7828548

CC(C)C[C@@H](C(=O)NN1C(=O)CN(CCN(C)C)C1=O)[C@H](CCCc1ccccc1)C(=O)NOCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 11/20 0.38
CTSK P43235 10/20 0.38
CTSB P07858 6/20 0.38
CTSS P25774 4/20 0.38
MMP1 P03956 1/20 0.38
MMP13 P45452 1/20 0.38
MMP3 P08254 1/20 0.34
ECE1 P42892 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7837319 1.00 CTSL (0.38) CTSLCTSKCTSBCTSSMMP1
SCHEMBL7955049 0.89 MMP1 (0.43) MMP1MMP13MMP3
SCHEMBL7836363 0.89 MMP1 (0.43) MMP1MMP13MMP3
SCHEMBL7955759 0.89 ACHE (0.36) CTSLCTSKCTSBCTSSMMP1
SCHEMBL7835837 0.89 ACHE (0.36) CTSLCTSKCTSBCTSSMMP1
SCHEMBL7953838 0.82 MMP1 (0.41) CTSLCTSKCTSBCTSSMMP1
SCHEMBL7841798 0.82 MMP1 (0.41) CTSLCTSKCTSBCTSSMMP1
SCHEMBL7946730 0.79 APP (0.49) MMP1MMP13MMP3
SCHEMBL7946731 0.79 APP (0.49) MMP1MMP13MMP3
SCHEMBL7846173 0.78 MMP1 (0.38) CTSLCTSKCTSBCTSSMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137640-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-10-04 EP disclosed
US-6281363-B1 ANTIINFLAMMATORY AGENTS; ANTIARTHRITIC AGENTS; AUTOIMMUNE DISORDERS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed
WO-2000035885-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-22 WO disclosed