SCHEMBL7828556

SCHEMBL7828556

CSc1ccc(C(C=O)c2cccc(F)c2)cc1C

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
ACHE P22303 1/20 0.33
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
ALDH1A1 P00352 1/20 0.31
AOC3 Q16853 1/20 0.31
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862422 0.80 HDAC4 (0.39) MEN1KMT2AHDAC4HDAC7HDAC5
SCHEMBL7917545 0.80 HDAC4 (0.47) HDAC4HDAC7HDAC5RAB9ACES2
SCHEMBL7029532 0.75 NPSR1 (0.34) MEN1KMT2AMAPT
SCHEMBL1515851 0.75 IDO1 (0.47) MEN1KMT2AHDAC4HDAC7HDAC5
SCHEMBL7861158 0.73 HDAC4 (0.42) HDAC4HDAC7HDAC5MAPTCES2
SCHEMBL7818627 0.71 AKR1C3 (0.44) CES2CES1
SCHEMBL3403146 0.70 CYP11B1 (0.41) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL7819110 0.70 SLC6A2 (0.34) MEN1KMT2AMAPTRAB9AIDO1
SCHEMBL8489218 0.69 ALDH1A1 (0.42) MEN1KMT2AMAPTRAB9ATAS1R3
SCHEMBL3905843 0.69 CES2 (0.44) HDAC4HDAC7HDAC5CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109799-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2001-06-27 EP disclosed
WO-2000061571-A1 4,5-DIARYL-3(2H)-FURANONE DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS PACIFIC CORPORATION (KR) 2000-10-19 WO disclosed