SCHEMBL7861158

SCHEMBL7861158

O=CC(c1ccc(Br)cc1)c1cccc(F)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
DPP4 P27487 1/20 0.36
HTR2A P28223 1/20 0.33
CNR2 P34972 1/20 0.33
NFE2L2 Q16236 1/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7917545 0.88 HDAC4 (0.47) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL1515851 0.86 IDO1 (0.47) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL7862422 0.81 HDAC4 (0.39) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL3403146 0.80 CYP11B1 (0.41) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL1515746 0.80 HTR2A (0.50) HTR2ACNR2SLC6A2SLC6A4
SCHEMBL4749525 0.80 CES2 (0.46) CES2MAPTIDO1TDO2SLC6A4
SCHEMBL7818627 0.78 AKR1C3 (0.44) CES2CES1
SCHEMBL2756356 0.76 ALDH1A1 (0.48) IDO1TDO2
SCHEMBL3905843 0.75 CES2 (0.44) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL931178 0.75 IDO1 (0.47) MAPTHTTIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086097-A1 SULFONYLBENZENE COMPOUNDS AS ANTI-INFLAMMATORY/ANALGESIC AGENTS PFIZER INC. (US) 2001-03-28 EP disclosed
WO-1999064415-A1 SULFONYLBENZENE COMPOUNDS AS ANTI-INFLAMMATORY/ANALGESIC AGENTS PFIZER PHARMACEUTICALS INC. (JP) 1999-12-16 WO disclosed