SCHEMBL7829862

SCHEMBL7829862

CCOC(=O)C1CN(CCC(=O)OCc2ccccc2)c2ccccc2O1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 11/20 0.49
KMT2A Q03164 1/20 0.45
SIRT2 Q8IXJ6 8/20 0.44
POLB P06746 1/20 0.44
ALDH1A1 P00352 2/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
P2RX1 P51575 1/20 0.41
P2RX3 P56373 1/20 0.41
P2RX4 Q99571 1/20 0.41
NOTUM Q6P988 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7819461 0.94 SIRT1 (0.47) SIRT1KMT2ASIRT2POLBALDH1A1
SCHEMBL7824177 0.90 ALDH1A1 (0.47) SIRT1KMT2APOLBALDH1A1TMEM97
SCHEMBL11567520 0.84 SIRT1 (0.69) SIRT1SIRT2POLB
SCHEMBL7809581 0.84 NOTUM (0.53) KMT2APOLBALDH1A1NOTUM
SCHEMBL7817475 0.84 SIRT1 (0.50) SIRT1KMT2ASIRT2POLBALDH1A1
SCHEMBL7817594 0.82 KMT2A (0.52) KMT2APOLBALDH1A1NOTUM
SCHEMBL8564037 0.81 P2RX4 (0.49) SIRT1KMT2APOLBALDH1A1P2RX1
SCHEMBL8564040 0.81 P2RX4 (0.49) SIRT1KMT2APOLBALDH1A1P2RX1
SCHEMBL8564035 0.81 P2RX4 (0.49) SIRT1KMT2APOLBALDH1A1P2RX1
SCHEMBL7820037 0.78 POLB (0.53) SIRT1KMT2ASIRT2POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894796-B1 Imidazolines substituted with a heterocyclic ring as alpha-2 antagonists ADIR (FR) 2001-06-06 EP disclosed
US-6057317-A Heterocyclic compounds ADIR ET COMPAGNIE (FR) 2000-05-02 US disclosed
EP-0894796-A1 Imidazolines substituted with a heterocyclic ring as alpha-2 antagonists ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed