SCHEMBL7830776

SCHEMBL7830776

CC(C)CCCOc1nsc(NC(=O)N(C)C)c1C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PPIA P62937 1/20 0.35
RARB P10826 1/20 0.33
MAPK1 P28482 1/20 0.32
C5 P01031 2/20 0.31
EPHX2 P34913 1/20 0.30
GPR88 Q9GZN0 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3094264 0.90 ACVR2A (0.36) PPIAC5
SCHEMBL3078154 0.86 ACVR2A (0.35) RARB
SCHEMBL7820761 0.83 LTA4H (0.41)
SCHEMBL7819943 0.81 KMT2A (0.44) MAPK1HPGD
SCHEMBL7831118 0.81 RARA (0.37) RARB
SCHEMBL7832137 0.77 GPR174 (0.33)
SCHEMBL7831489 0.77 NR3C2 (0.40) HPGD
SCHEMBL3071384 0.75 XDH (0.38)
SCHEMBL3093008 0.74 ACVR2A (0.36)
SCHEMBL3087282 0.74 MEN1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1084114-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2001-03-21 EP disclosed
WO-1999062890-A1 ISOTHIAZOLE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-12-09 WO disclosed