SCHEMBL7832205

SCHEMBL7832205

COc1ccccc1N1CCN(CCCn2c(=O)c(C)cn(C)c2=O)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.60
KMT2A Q03164 3/20 0.60
DRD2 P14416 2/20 0.59
DRD3 P35462 2/20 0.59
HTR1A P08908 7/20 0.59
HTR7 P34969 7/20 0.59
ADRA2A P08913 2/20 0.58
ADRA2B P18089 2/20 0.58
ADRA2C P18825 2/20 0.58
ADRB2 P07550 1/20 0.58
CYP1A2 P05177 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
ADRA1B P35368 3/20 0.57
CYP3A4 P08684 2/20 0.57
ADRA1D P25100 2/20 0.57
ADRA1A P35348 2/20 0.57
HIF1A Q16665 2/20 0.57
PMP22 Q01453 1/20 0.57
HTR2A P28223 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7832997 0.99 MEN1 (0.59) MEN1KMT2ADRD2DRD3HTR1A
SCHEMBL7830329 0.86 HTR1A (0.56) MEN1KMT2ADRD2DRD3HTR1A
Hydrochloric Acid SCHEMBL7833555 0.85 ADRA1A (0.71) CYP2C9CYP2C19ADRA1BCYP3A4ADRA1D
Hydrochloric Acid SCHEMBL7821236 0.85 HTR1A (0.55) MEN1KMT2ADRD2DRD3HTR1A
Hydrochloric Acid SCHEMBL7832683 0.83 HTR1A (0.62) MEN1KMT2ADRD2DRD3HTR1A
SCHEMBL7834491 0.82 HTR1A (0.56) DRD2DRD3HTR1AHTR7ADRA2A
SCHEMBL7836830 0.82 ADRA1A (0.75) MEN1KMT2ADRD2DRD3HTR1A
Hydrochloric Acid SCHEMBL7834012 0.81 HTR1A (0.55) DRD2DRD3HTR1AHTR7ADRA2A
Hydrochloric Acid SCHEMBL7830482 0.81 ADRA1A (0.74) MEN1KMT2ADRD2DRD3HTR1A
SCHEMBL6526368 0.81 DRD2 (0.85) MEN1KMT2ADRD2DRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748800-B1 Pyrimidinedione, pyrimidinetrione, triazinedione derivatives as alpha-1-adrenergic receptor antagonists HOFFMANN LA ROCHE (CH) 2001-05-09 EP disclosed
EP-0748800-A2 Pyrimidinedione, pyrimidinetrione, triazinedione, tetrahydroquinazolinedione derivatives as alpha-1-adrenergic receptor antagonists F. HOFFMANN-LA ROCHE AG (CH) 1996-12-18 EP disclosed